目錄:MedChemExpress LLC>>生化試劑>> Tacrine hydrochloride (hydrate) | MCE
CAS | 206658-92-6 | 純度 | 99.98% |
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分子式 | C??H??N?.xHCl.xH?O | 供貨周期 | 現貨 |
規格 | 100 mg | 貨號 | HY-B2244 |
應用領域 | 醫療衛生,化工,生物產業,制藥 |
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CAS No. : 206658-92-6
產品活性:Tacrine hydrochloride (hydrate) is an inhibitor of both acetyl (AChE) and butyryl-cholinestrase (BChE) with IC50s of 31 nM and 25.6 nM, respectively.
研究領域:Neuronal Signaling
作用靶點:Cholinesterase (ChE)
In Vitro: Tacrine hydrochloride (hydrate) (12.5 to 37.5 nM) inhibits venom acetylcholinesterase as well as human serum butyrylcholinesterase in a concentration-dependent manner. The IC50 is 31 nM for snake venom AChE and 25.6 nM for human BChE.
In Vivo: Pretreatment with Tacrine hydrochloride (hydrate) also modifies absolute levels of cocaine self-administration during reacquisition. Body weight declines approximately one-half percent over four days of treatment with intravenous Tacrine hydrochloride (hydrate). Delivery of Tacrine hydrochloride (hydrate) by osmotic pump does not alter either linear- or repeated- cocaine-induced locomotor activity. There is no significant main effect or interaction with Tacrine hydrochloride (hydrate) treatment on active lever responding during reinstatement. Post hoc comparisons indicate that rats self-administering cocaine has significantly lower alkaline phosphatase levels, relative to TTacrine hydrochloride (hydrate)- but not saline- treated rats evaluated by conditioned-place preference.
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